| 2OG | 2-Oxoglutarate |
| ATP | Adenosine triphosphate |
| DCC | Dynamic combinatorial chemistry |
| DCL | Dynamic combinatorial library |
| DNA | Deoxyribonucleic acid |
| FITC | Fluorescein isothiocyanate |
| GABA | γ-Animobytyric acid |
| GAT1 | γ-Animobytyric acid transporter 1 |
| HEWL | Hen egg-white lysozyme |
| HIF | Hypoxia inducible factor |
| HPLC | High-performance liquid chromatography |
| HSP | Heat shock protein |
| HTS | High-throughput screening |
| JMJD2 | Jumonji domain 2 |
| LC-MS | Liquid chromatography-mass spectrometry |
| NMR | Nuclear magnetic resonance |
| NOE | Nuclear Overhauser effect |
| PHD2 | Prolyl hydroxylase domain 2 |
| STD | Saturation transfer difference |
| TPR | Tetratricopeptide repeat |
| WaterLOGSY | Water ligand-observed via gradient spectroscopy |