Figure 1.
Structure and affinities of 5-HT6R ligands. Agonists: 5-HT and 2-Me 5-HT, Antagonists: LSD, Clozapine and N-arylsulfonylindole I to VI. (Ki = inhibitory constant from radioligand binding assays, see Section 4.5).
Structure and affinities of 5-HT6R ligands. Agonists: 5-HT and 2-Me 5-HT, Antagonists: LSD, Clozapine and N-arylsulfonylindole I to VI. (Ki = inhibitory constant from radioligand binding assays, see Section 4.5).