Table 3.
Acid | Equivalents of amine | Yield of isolated product [%] |
---|---|---|
6 | 2 | 85 (6 a) |
10 | 2 | 70 (10 a)[a] |
14 | 2 | 50 (14 a) |
16 | 5 | 15 (16 a) |
17 | 5 | 51 (17 a) |
19 | 5 | 21 (19 a) |
[a] carried out on 30 mg scale
Acid | Equivalents of amine | Yield of isolated product [%] |
---|---|---|
6 | 2 | 85 (6 a) |
10 | 2 | 70 (10 a)[a] |
14 | 2 | 50 (14 a) |
16 | 5 | 15 (16 a) |
17 | 5 | 51 (17 a) |
19 | 5 | 21 (19 a) |
[a] carried out on 30 mg scale