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. 2018 Nov 29;9(12):1292–1296. doi: 10.1021/acsmedchemlett.8b00504

Table 1. Equilibrium and Kinetic Constants of PE2I and FE-PE2I Binding to DAT.

compd Ki, nM KL, nM ki, min–1 k–i, min–1 Kisom
FE-PE2I 23 ± 3 79 ± 33 0.34 ± 0.06 0.15 ± 0.09 0.44
PE2Ia 5 ± 1 37 ± 24 1.2 ± 0.5 0.14 ± 0.05 0.12
a

Data from ref (20).