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Inhibition potency of hASIC3 antagonists.
| Antagonist | Transient Currents | Sustained Currents | ||
|---|---|---|---|---|
| IC50 (µM) | Hill Coefficient | IC50 (µM) | Hill Coefficient | |
| APETx2 | 0.344 ± 0.080 | 1.5 ± 0.2 | - | - |
| Ugr 9-1 | 9.1 ± 0.9 | 1.86 ± 0.16 | 1.88 ± 0.36 | 1.74 ± 0.51 |
| sevanol | 331 ± 21 | 1.98 ± 0.24 | 259 ± 39 | 2.4 ± 0.4 |
| diclofenac | - | - | 856 ± 106 | 1.35 ± 0.21 |
