Table 2.
Whole cell HDAC enzyme inhibition assay.
| Sl. no. | Compound | HDAC inhibition IC50 (µM ± SEM) |
|---|---|---|
| 1 | QMJ-1 | 1023.1 ± 5.2 |
| 2 | QMJ-2 | 181.7 ± 22.04 |
| 3 | QMJ-3 | 1124 ± 6.2 |
| 4 | QMJ-4 | 1011.2 ± 3.4 |
| 5 | QMJ-5 | 70.2 ± 4.3 |
| 6 | QMJ-6 | 984.2 ± 2.5 |
| 7 | Quercetin | 167.8 ± 6.9 |
| 8 | SAHA | 1.2 ± 0.1 |
The values are expressed as mean ± SEM of three experiments.