Table 3. Potency (EC50, μM) of RTG, 8g, 10g, and 13 against KCNQ4, KCNQ5, and KCNQ2.
RTG | 8g | 10g | 13 | |
---|---|---|---|---|
KCNQ4 | 5.90 ± 0.18 | 2.03 ± 0.14 | 0.78 ± 0.14 | 1.42 ± 0.04 |
KCNQ5 | 3.45 ± 0.28 | 2.43 ± 0.17 | 1.68 ± 0.12 | 1.37 ± 0.11 |
KCNQ2 | 2.17 ± 0.07 | >30 | >30 | >30 |