Scheme 2. Results for the Suzuki–Miyaura Cross Coupling of 8 with an Informer Library of Pinacol Boronate Esters.
Yields listed are based on 19F NMR spectroscopic analysis of 0.010 mmol scale screening reactions. Isolated yields of 0.1–0.4 mmol scale reactions are listed in parentheses (see SI for details).