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. Author manuscript; available in PMC: 2019 Jan 22.
Published in final edited form as: Curr Pharm Des. 2014;20(5):793–807. doi: 10.2174/138161282005140214165212

Table 3.

Common drugs transported by P-gp, MRP1 and BCRP.

P-gp (ABCB1) Anticancer drues: doxorubicin, daunorubicin. epirubicin. colchicine, antinomvcin D. etoposide. teniposide. methotrexate, mitocvcin C, paclitaxel, mitoxantrone, docetaxel, vinblastine, vincristine
Antihvnertensives: losartan. celiorolol. reseroine. talinolol. Nicardipine
Antiarrhvthimics: dieoxin. propafenone, auinidine. verapamil, amiodarone
Antibiotics: ervthromvcin. rifampin, levofloxacin. clarithromycin, tetracycline
Antivirals: amorenavir. indinavir, nelfinair. ritonavir, saauinavir
Antidepressants: amitrintvline. fluoxetine, paroxetine, sertraline
Immunosuppressants: cyclosporine A. sirolimus. tacrolimus, valspodar
Opioids: methadone, morphine
Lipid lowerine drues: atorvastatin. lovastatin
Glucocorticoids: aldosterone, cortisol, dexamethasone. Methvlprednisolone
Antihistamines: fexofenadine, terfenadine
Others: oroeesterone. itraconazole, phenobarbital. phenvtoin. cimetidine
MRP1 (ABCC1) Anticancer drues: doxorubicin, daunorubicin. colchicine, toootecan. irinotecan. SN-38. methotrexate, etoposide. teniposide. vincristine.
vinblastine, imatinib, gefitinib
Antivirals: indinavir, ritonavir, saauinavir
Antibiotics: ciprofloxacin, difloxacin. ereoafloxacin. pirarbicin
BCRP (ABCG2) Anticancer drues: doxorubicin, daunorubicin. epirubucin. methotrexate, toootecan. irinotecan, SN-38. etoposide. teniposide. imatinib, gefitinib
Antibiotics: ciprofloxacin, norfloxacin, ofloxacin
Lipid lowerine drues: cerivastatin. pravastatin, rosuvastatin
Antivirals: lamivudine. Zidovudine
Antihvoertensives: reseroine
Others: azidothvmidine. lamivudine