Table 3.
Common drugs transported by P-gp, MRP1 and BCRP.
P-gp (ABCB1) | Anticancer drues: doxorubicin, daunorubicin. epirubicin. colchicine, antinomvcin D. etoposide. teniposide. methotrexate, mitocvcin C, paclitaxel, mitoxantrone, docetaxel, vinblastine, vincristine |
Antihvnertensives: losartan. celiorolol. reseroine. talinolol. Nicardipine | |
Antiarrhvthimics: dieoxin. propafenone, auinidine. verapamil, amiodarone | |
Antibiotics: ervthromvcin. rifampin, levofloxacin. clarithromycin, tetracycline | |
Antivirals: amorenavir. indinavir, nelfinair. ritonavir, saauinavir | |
Antidepressants: amitrintvline. fluoxetine, paroxetine, sertraline | |
Immunosuppressants: cyclosporine A. sirolimus. tacrolimus, valspodar | |
Opioids: methadone, morphine | |
Lipid lowerine drues: atorvastatin. lovastatin | |
Glucocorticoids: aldosterone, cortisol, dexamethasone. Methvlprednisolone | |
Antihistamines: fexofenadine, terfenadine | |
Others: oroeesterone. itraconazole, phenobarbital. phenvtoin. cimetidine | |
MRP1 (ABCC1) |
Anticancer drues: doxorubicin, daunorubicin. colchicine, toootecan. irinotecan. SN-38. methotrexate, etoposide. teniposide. vincristine. vinblastine, imatinib, gefitinib |
Antivirals: indinavir, ritonavir, saauinavir | |
Antibiotics: ciprofloxacin, difloxacin. ereoafloxacin. pirarbicin | |
BCRP (ABCG2) | Anticancer drues: doxorubicin, daunorubicin. epirubucin. methotrexate, toootecan. irinotecan, SN-38. etoposide. teniposide. imatinib, gefitinib |
Antibiotics: ciprofloxacin, norfloxacin, ofloxacin | |
Lipid lowerine drues: cerivastatin. pravastatin, rosuvastatin | |
Antivirals: lamivudine. Zidovudine | |
Antihvoertensives: reseroine | |
Others: azidothvmidine. lamivudine |