Table 3. The structures of six newly designed compounds and their activity against DENV-2 NS2B/NS3pro.
Ligands | R1 | R2 | R3 | IC50 (μM) |
---|---|---|---|---|
16 | propanoyl | propanoyl | H | 97 |
17 | isopropanoyl | isopropanoyl | H | 80 |
18 | pentanoyl | pentanoyl | H | 0.38 |
19 | pentanoyl | benzyl | H | 54 |
20 | H | 2-methylnaphtyl | isopropyl | 258 |
21 | pentanoyl | benzyl | benzyl | 16 |