Table 1.
CYP2D6 inhibitors observed in study, by inhibitor strength and exposure classification
Exposure classification | ||||
---|---|---|---|---|
Strength | Medications | Any inhibition |
Strong or moderate |
Strong only |
Strong | bupropion, fluoxetine, paroxetine | X | X | X |
Moderate | duloxetine, sertraline | X | X | |
Weak or unknown | amiodarone, celecoxib, citalopram, clomipramine, diltiazem, doxepin, escitalopram, hydralazine, oral contraceptives, propafenone, verapamil | X |