Table 1.
Kinetic parameters for BPAF glucuronidation by UGTs 1A3, 1A10, 2A1, 2B7, and 2B17.
| Enzyme | Model | Vmax(nmol/min/mg) | Km(µM) | r2 | Ksi |
|---|---|---|---|---|---|
| 2A1 | MM | 3.3 ± 0.1 | 8.4 ± 0.8 | 0.98 | |
| 1A10 | SI | 3.0 ± 0.4 | 18 ± 3 | 0.99 | 35 ± 8 |
| 2B7 | SI | 0.21 ± 0.01 | 0.9 ± 0.1 | 0.96 | 27 ± 3 |
| 2B17 | SI | 0.33 ± 0.01 | 1.1 ± 0.1 | 0.98 | 123 ± 25 |
| 1A3 | SI | 0.79 ± 0.17 | 22 ± 6 | 0.98 | 8.0 ± 2.1 |