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. Author manuscript; available in PMC: 2019 Feb 1.
Published in final edited form as: Chem Rev. 2016 Oct 19;117(4):2711–2729. doi: 10.1021/acs.chemrev.6b00400

Table 3.

Comparison of IC50 cytotoxicity values of 1-Ga, Ga(ACtpfc) and Ga(3-ctpfc) in human cancer cell lines. Reproduced from ref. 114. Copyright 2016 National Academy of Sciences.

Cell line DU145 SK-MEL-28 MDA-MB-231 OVCAR-3
Tumor type prostate Melanoma breast ovarian
IC50 (µM) 1-Ga 158.9 131.4 129.2 274.2
Ga(ACtpfc) 17.6 14.4 13.7 12.7
Ga(3-ctpfc) 12.9 4.8 15.3 11.1