Table 2. Structure–Activity Relationship of Linker Moiety1.
i.a., inactive at 30 μM; relative activation efficacy compared to 1 (1 μM) is shown in parentheses. All values are mean ± SEM; n ≥ 3.
i.a., inactive at 30 μM; relative activation efficacy compared to 1 (1 μM) is shown in parentheses. All values are mean ± SEM; n ≥ 3.