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. 2019 Jan 4;10(2):203–208. doi: 10.1021/acsmedchemlett.8b00551

Table 4. Combinations of Structural Motifs for Enhanced Potency Identified in SAR Studies1.

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1

tox., toxic at 30 μM; relative activation efficacy compared to 1 (1 μM) is shown in parentheses. All values are mean ± SEM; n ≥ 3.