Skip to main content
. 2019 Jan 15;10(2):268–279. doi: 10.1039/c8md00405f

Table 3. Group II click products 46–57 of halogenated azidomethylsulfoxides 11, 12 and azidophenyl sulfones 14, 15 with selected arylacetylenes 17–19.

Inline graphic
Compound Yield a (%)
46, R1 = 4-fluorophenyl, R2 = 3-fluorophenyl, R3 = SO 78
47, R1 = 4-fluorophenyl, R2 = 4-fluorophenyl, R3 = SO 83
48, R1 = 4-fluorophenyl, R2 = 2-methoxypheny, R3 = SO 92
49, R1 = 4-chlororophenyl, R2 = 3-fluorophenyl, R3 = SO 52
50, R1 = 4-chlorophenyl, R2 = 4-fluorophenyl, R3 = SO 93
51, R1 = 4-chlorophenyl, R2 = 2-methoxyphenyl, R3 = SO 76
52, R1 = 4-fluorophenyl, R2 = 3-fluorophenyl, R3 = SO2 79
53, R1 = 4-fluorophenyl, R2 = 4-fluorophenyl, R3 = SO2 83
54, R1 = 4-fluorophenyl, R2 = 2-methoxyphenyl, R3 = SO2 95
55, R1 = 4-chlororophenyl, R2 = 3-fluorophenyl, R3 = SO2 84
56, R1 = 4-chlorophenyl, R2 = 4-fluorophenyl, R3 = SO2 93
57, R1 = 4-chlorophenyl, R2 = 2-methoxyphenyl, R3 = SO2 81

aYields are for isolated pure compounds.