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. 2018 Dec;56(4):553–561. doi: 10.17113/ftb.56.04.18.5553

Table 1. Effects of specific inhibitors on the protease activity.

    c(inhibitor)/mM     Residual activity/%
    0.1     1
    None     100     100
    DFP     10     5
    Pefabloc     18     9
    PMSF     40     25
    EDTA     99     95
    EGTA     90     90
    1,10-Phenanthroline     100     95
    Iodoacetamide     100     100
    E-64     100     100
    Pepstatin A     100     100
    10–3     10–2
    Bestatin     100     100
    TLCK     100     100
    10–4     10–3
    Aprotinin     100     100

DFP=diisopropyl fluorophosphates, PMSF=phenylmethylsulfonyl fluoride, EDTA=ethylenediaminetetraacetic acid, EGTA=ethylene-bis(oxyethylenenitrilo)tetraacetic acid tetrasodium, TLCK= Nα-tosyl--l-lysine chloromethyl ketone hydrochloride