Skip to main content
. Author manuscript; available in PMC: 2019 Apr 17.
Published in final edited form as: Chem Rev. 2018 Sep 7;119(2):1323–1455. doi: 10.1021/acs.chemrev.8b00201

Table 9.

Activity of LF inhibitors.

Compound Inhibition (μM) Ref.
LFi-1 Ki = 0.001 616
LFi-2 Ki = 2.1 617
LFi-3 Ki = 0.024 618
LFi-4 Ki = 0.00031 620
LFi-5 Ki = 0.00027 620
LFi-6 IC50 = 1.6 622
LFi-7 IC50 = 5.6 622
LFi-8 IC50 = 4.4 622
LFi-9 IC50 = 1.4 619
LFi-10 Ki = 0.0014 626
LFi-11 Ki = 0.0064 626
LFi-12 Ki = 3 627
LFi-13 Ki > 100 627
LFi-14 Ki > 100 627
LFi-15 Ki = 1.7 627
LFi-16 IC50 = 70 627
LFi-17 Ki = 6.0 627
LFi-18 IC50 ~2 628
LFi-19 IC50 = 50 628
LFi-20 IC50 = 260 629
LFi-21 IC50 >6000 629
LFi-22 IC50 = 13.9 629
LFi-23 IC50 = 5.0 630
LFi-24 IC50 = 15 621
LFi-25 IC50 = 21 621
LFi-26 IC50 > 100 621
EGCG IC50 = 0.097 631