Table 2.
Structure-activity analysis of substituted phenol compounds.
Compound | IC50 (μM) | Estimated Vapor Pressure (mmHg at 25 °C) | Boiling Point (degrees C) |
---|---|---|---|
![]() |
15 ± 1 | 0.003 | 281.2 |
![]() |
25 ± 3 | 0.01 | 247.7 |
![]() |
32 ± 5 | 0.05 | 229.7 |
![]() |
37 ± 7 | 0.003 | 261.4 |
![]() |
50 ± 7 | 0.001 | 271.4 |
![]() |
86 ± 17 | 0.008 | 247.7 |
![]() |
92 ± 9 | 0.007 | 281.2 |
![]() |
212 ± 29 | 0.02 | 229.6 |
![]() |
261 ± 14 | 0.15 | 210.7 |
IC50 values for inhibition of Agam\Orco are presented as mean ± SEM (n = 3–9). Vapor pressures and boiling points were estimated as described in Methods.