Table 3.
Number of unique compounds with categorigal activity annotations from the open domain.
Transporter | UNIPROT ID | Metrabase | Drugbank | Total number of unique compounds |
---|---|---|---|---|
OCT1 | O15245 | 504 | 69 | 470 |
OCT2 | O15244 | No entries | 56 | 56 |
OCT3 | O75751 | No entries | 29 | 29 |
OCTN1 | Q9H015 | No entries | 27 | 27 |
OCTN2 | O76082 | No entries | 54 | 54 |
MATE1 | Q96FL8 | No entries | 6 | 6 |
MATE2-K | Q86VL8 | No entries | 1 | 1 |
OAT1 | Q4U2R8 | No entries | 111 | 111 |
OAT2 | Q9Y694 | No entries | 36 | 36 |
OAT3 | Q8TCC7 | No entries | 77 | 77 |
OATP1B1 | Q9Y6L6 | 375 | 75 | 385 |
OATP1B3 | Q9NPD5 | 338 | 44 | 345 |
OATP1A2 | P46721 | 111 | 61 | 107 |
OATP2B1 | O94956 | 352 | 33 | 338 |