Table 3.
LDA inhibitory activity and cytotoxicity
Nos. | LDA inhibitory IC50 (μM) | Cytotoxicity CC50 (μM) | Selectivity index (CC50/IC50) |
---|---|---|---|
1 | 11.6 | 29.4 | 2.5 |
2 | 7.1 | >50 | >7.0 |
3 | 3.3 | >50 | >15.2 |
4 | >50 | >50 | ND |
5 a | 1.8 | 15.9 | 8.8 |
6 | 4.7 | 53.2 | 11.3 |
7 | 12.2 | >50 | >4.1 |
8 | >50 | >50 | ND |
9 | 11.6 | 18.3 | 1.6 |
10 | 12.0 | 18.9 | 1.6 |
11 | 14.8 | >50 | >3.4 |
12 a,b | 8.8 | 26.2 | 3.0 |
13 a,c | 7.7 | 20.6 | 2.7 |
14 a,d | >50 | >50 | ND |