Table 3.
LDA inhibitory activity and cytotoxicity
| Nos. | LDA inhibitory IC50 (μM) | Cytotoxicity CC50 (μM) | Selectivity index (CC50/IC50) |
|---|---|---|---|
| 1 | 11.6 | 29.4 | 2.5 |
| 2 | 7.1 | >50 | >7.0 |
| 3 | 3.3 | >50 | >15.2 |
| 4 | >50 | >50 | ND |
| 5 a | 1.8 | 15.9 | 8.8 |
| 6 | 4.7 | 53.2 | 11.3 |
| 7 | 12.2 | >50 | >4.1 |
| 8 | >50 | >50 | ND |
| 9 | 11.6 | 18.3 | 1.6 |
| 10 | 12.0 | 18.9 | 1.6 |
| 11 | 14.8 | >50 | >3.4 |
| 12 a,b | 8.8 | 26.2 | 3.0 |
| 13 a,c | 7.7 | 20.6 | 2.7 |
| 14 a,d | >50 | >50 | ND |