Table 2. In Vitro Pharmacokinetics for Compounds 3f and 13.
compound | solubilitya (μM) | log D | Clintb | t1/2 (min) | %c |
---|---|---|---|---|---|
3f | 200 | 0.34 | 20.67 | 111.8 | 76.2 |
13 | 110.4 | 0.58 | 201 | 11.5 | 9.4 |
Aqueous solubility at pH 7.4.
Reported as μL/min/mg protein.
Percentage of compound remaining in solution after 40 min of incubation. Each measurement has been repeated in triplicate and SD < 5%.