Table 2. Pharmacokinetic parameters of aniracetam and N-anisoyl-GABA following oral administration of aniracetam to pigeons.
Pharmacokinetic parameter | Aniracetam | N-anisoyl-GABA |
---|---|---|
100 mg/kg | ||
AUClast (ng·h/mL) | 9,309.62 | 173,740 |
AUMC (ng·h2/mL) | 274,098.78 | 8,633,225 |
Cmax (ng/mL) | 242.96 | 4,254.87 |
Tmax (min) | 15 | 10 |
MRT (h) | 29.44 | 49.69 |
200 mg/kg | ||
AUClast (ng·h/mL) | 74,927 | 311,055 |
AUMC (ng·h2/mL) | 4,082,985 | 1.9 x 107 |
Cmax (ng/mL) | 1,463.60 | 6379.44 |
Tmax (min) | 90 | 90 |
MRT (h) | 54.49 | 60.88 |