Table 2. KiNativ™ assay tests for SAB298 target protein*.
Kinase | YUSIV | YUSIK |
---|---|---|
YES1 | <10 | Not Present |
SRC | 31 | Not Present |
LYN | 60 | 190 |
ABL2 | 87 | 240 |
ERBB3 | 290 | 240 |
MEK5 | 370 | 1500 |
CSK | 420 | 910 |
ERBB2 | 410 | 530 |
mTOR | 1,300 | 2,000 |
EGFR | 1,300 | 530 |
LCK | 1,400 | Not Present |
RIPK2 | Not Present | 20 |
MEK1 | 2,900 | Not Present |
*The results show IC50 in nM. Values were determined from 3-point dose response curve.