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. 2019 Mar;16(3):182–241. doi: 10.11909/j.issn.1671-5411.2019.03.014

Table 9. Single-pill combination preparations.

Major components and single dose Tablets per day Times per day Major side effects
Losartan pot./Hydrochlorothiazide Angioneurotic edema (occasional) and abnormal serum potassium
 50 mg/12.5 mg 1 1
 100 mg/12.5 mg 1 1
 100 mg/25 mg 1 1
Valsartan/Hydrochlorothiazide Angioneurotic edema (occasional) and abnormal serum potassium
 80 mg/12.5 mg 1–2 1
Irbesartan/Hydrochlorothiazide 1 1 Angioneurotic edema (occasional) and abnormal serum potassium
 150 mg/12.5 mg
Telmisartan/Hydrochlorothiazide 1 1 Angioneurotic edema (occasional) and abnormal serum potassium
 40 mg/12.5 mg
 80 mg/12.5 mg 1 1
Olmesartan/Hydrochlorothiazide 1 1 Angioneurotic edema (occasional) and abnormal serum potassium
 20 mg/12.5 mg
Captopril/Hydrochlorothiazide 1–2 1–2 Coughing, angioneurotic edema (occasional), abnormal serum potassium
 10 mg/6 mg
Lisinopril/Hydrochlorothiazide 1 1 Coughing, angioneurotic edema (occasional), abnormal serum potassium
 10 mg/12.5 mg
Enalapril/Hydrochlorothiazide 1 1 Coughing, angioneurotic edema (occasional), abnormal serum potassium
 5 mg/12.5 mg
Benazepril/Hydrochlorothiazide 1 1 Coughing, angioneurotic edema (occasional), abnormal serum potassium
 10 mg/12.5 mg
Perindopril/Indapamide 1 1 Coughing, angioneurotic edema (occasional), abnormal serum potassium
 4 mg/1.25 mg
Perindopril/Amlodipine 1 1 Dizziness, headache and coughing
 10 mg/5 mg
Amlodipine/Valsartan 1 1 Headache, ankle edema, angioneurotic edema (occasional)
 5 mg/80 mg
Amlodipine/Telmisartan 1 1 Headache, ankle edema, angioneurotic edema (occasional)
 5 mg/80 mg
Amlodipine/Benazepril 1 1 Headache, ankle edema, angioneurotic edema (occasional)
 5 mg/10 mg
 2.5 mg/10 mg 1 1 Headache, ankle edema, angioneurotic edema (occasional)
Amiloride/Hydrochlorothiazide 1 1 Abnormal serum potassium, hyperuricemia
 2.5 mg/25 mg
Nitrendipine/Atenolol 1 1–2 Headache, ankle edema, bronchospasm, bradycardia
 10 mg/20 mg
 5 mg/10 mg 1–2 1–2
Reserpine/Hydrochlorothiazide/Dihydralazine/Promethazine 1–3 2–3 Digestive ulceration and sleepiness
 0.032 mg/3.1 mg/4.2 mg/2.1 mg
Reserpine/Triamterene Hydrochlorothiazide/Dihydralazine 1–2 1 Digestive and headache
 0.1 mg/12.5 mg/12.5 mg/12.5 mg
Zhenjujiangya tablet 1–3 2–3 Hypotension and abnormal serum potassium
 Clonidipine 0.03 mg/Hydrochlorothiazide 5 mg
Enalapril/Folic acid 1–2 1–2 Coughing, nausea, angioneurotic edema (occasional), headache, ankle edema, myalgia
 10 mg/0.8 mg
Amiloride/Atorvastatin 1 1 Transaminase elevation
 5 mg/10 mg
Candesartan/Hydrochlorothiazide 1 1 Upper respiratory tract infection, backache, abnormal serum potassium
 16 mg/12.5 mg

For details on the usage of antihypertensive drugs, please refer to the relevant manual approved by China Food and Drug Administration.