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| assay | value |
|---|---|
| solubility (CLND) | 119 μM |
| CHROM LogD (pH 7.4) | 3.6 |
| artificial membrane permeability | 2.1 × 10–5 cm/s |
| fraction bound in blood (mouse, rat, human) | 99.5%, 99.6%, 99.3% |
| microsomal clearance (mouse, rat, human) | 8.5, 2.1, 1.1 mL/min/g tissue |
| microsomal half-life (mouse, rat, human) | 8.5, 34.2, 67.4 min |
