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. 2017 Oct 3;21(6):805–812. doi: 10.1093/ntr/ntx187

Table 1.

Responses of nAChR Subtypes to 100 μM DMPA Relative to ACh Maximum Response

α4(3)β2(2) 0.47 ± 0.12
α4(2)β2(3) 0.46 ± 0.05
α4(2)β2(2)α5 0.39 ± 0.02
α6β2β3α4β2 0.46 ± 0.01
α3β4 0.01 ± 0.00
α1β1εδ 0.40 ± 0.03
α7 0.41 ± 0.02
α7a 20.83 ± 5.29

aNet charge response to 100 μM 4-acetyl-1,1-dimethylpiperazin-1-ium plus 10 μM PNU-120596 relative to acetylcholine alone.

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