Table 1.
Responses of nAChR Subtypes to 100 μM DMPA Relative to ACh Maximum Response
α4(3)β2(2) | 0.47 ± 0.12 |
α4(2)β2(3) | 0.46 ± 0.05 |
α4(2)β2(2)α5 | 0.39 ± 0.02 |
α6β2β3α4β2 | 0.46 ± 0.01 |
α3β4 | 0.01 ± 0.00 |
α1β1εδ | 0.40 ± 0.03 |
α7 | 0.41 ± 0.02 |
α7a | 20.83 ± 5.29 |
aNet charge response to 100 μM 4-acetyl-1,1-dimethylpiperazin-1-ium plus 10 μM PNU-120596 relative to acetylcholine alone.