Concentration-dependent effect of reference A3AR agonist
2-Cl-IB-MECA on βarr2 recruitment in a stable
hA3AR-NanoBit®-βarr2 HEK293T cell line.
1, 2, 5, 10, 30, 50, 80, 100, 500 nM and 1 µM 2-Cl-IB-MECA was added at
the time point indicated by the arrow, and luminescence was measured for
>90 min. A solvent control of 0.01% DMSO was included. Insert:
Concentration-response (AUCs). AUCs (± SEM) of quadruplicate wells are
shown for a representative experiment (n=3).