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. Author manuscript; available in PMC: 2020 Jan 24.
Published in final edited form as: J Med Chem. 2018 Dec 10;62(2):448–466. doi: 10.1021/acs.jmedchem.8b00909

Figure 1.

Figure 1.

(A) Co-crystal structure of MDM2 in a complex with MI-77301 (Cyan), (PDB ID: 5TRF); (B) Modeled structure of MDM2 complexed with MI-1061 (Yellow); (C) Chemical structures of MDM2 inhibitors MI-77301 and MI-1061.