Table 4.
entry | product, R1, R2 | yield (%)b |
---|---|---|
1 | 6a, Ph, Me | 60 |
2 | 6b, Ph, n-C6H13 | 66 |
3 | 6c, Ph, Cy | 51 |
4 | 6d, Ph, CF3 | 60 |
5 | 6e, Cy, Me | 82 |
Reactions under N2 with 0.2 mmol of tetrahydroisoquinoline (0.8 M).
Isolated yields of purified products.