Table 2. Lead Compound 9 to Candidate Compound 11a.
Footnote: *Activity screen assay linearity from 0.01 to 10 μM. Values are mean ± SD. Values outside linearity, >10 μM. Human liver microsome assay, linear to 60 min.
Footnote: *Activity screen assay linearity from 0.01 to 10 μM. Values are mean ± SD. Values outside linearity, >10 μM. Human liver microsome assay, linear to 60 min.