. 2019 Apr 29;29(7):530–542. doi: 10.1093/glycob/cwz029

Table I.

Inhibition data of four active compounds towards ER α-Glu II as determined by a calorimetric kinetic assay using purified GIIα

Compound	Inhibition Mode	K_i (μM)^a	K_i (μM)^b
DAB	Competitive	0.187 ± 0.003	0.170 ± 0.003
CST	Competitive	2.60 ± 0.58	3.15 ± 0.10
CSU	Competitive	4.07 ± 0.06	4.15 ± 0.056
DMDP	Competitive	18.07 ± 0.51	14.95 ± 0.60

^aK_i was calculated using K_M and V_MAX values obtained from controls (n = 3) per compound

^bK_i was calculated using K_M and V_MAX values obtained from controls (n = 12) across all four compounds