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. Author manuscript; available in PMC: 2020 Apr 3.
Published in final edited form as: J Am Chem Soc. 2019 Mar 21;141(13):5135–5138. doi: 10.1021/jacs.9b01091

Table 3.

Scope of DKR E-CuAAC with Respect to Azide 1

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Yields are reported for isolated and purified products. Enantiomeric ratio was determined by chiral HPLC. Yield and er values reflect the average of duplicate trials.

a

Reaction used alkyne as limiting reagent. See Supporting Information for details.