Table 1.
Agonists and antagonists of TRPV
| TRPV1 |
TRPV2 |
TRPV3 |
TRPV4 |
Other TRPs |
References | ||||||
|---|---|---|---|---|---|---|---|---|---|---|---|
| Agonist | Antagonist | Agonist | Antagonist | Agonist | Antagonist | Agonist | Antagonist | Agonist | Antagonist | ||
| Lanthanum | — | + | — | + | — | + | — | + | — | + | (Wu et al., 2010) |
| Gadolinium | — | + | — | + | — | + | — | + | — | + | |
| Ruthenium red | — | + | — | + | — | + | — | + | — | + | |
| FFA | — | + | — | + | — | + | — | + | — | + | (Guinamard et al., 2013) |
| 2APB | + | — | + | — | + | — | — | — | — | + | (Hu et al., 2004; Harteneck and Gollasch, 2011) |
| SKF 96365 | — | — | — | — | — | — | — | — | — | + | (Wu et al., 2010) |
| Capsaicin | + | — | — | — | — | — | — | — | — | — | (Caterina et al., 1997) |
| Capsazepine | — | + | — | — | — | — | — | — | — | — | (Caterina et al., 1997) |
| Probenecid | — | — | + | — | — | — | — | — | — | — | (Bang et al., 2007) |
| Tranilast | — | — | — | + | — | — | — | — | — | — | (Hisanaga et al., 2009) |
| Camphor | — | — | — | — | + | — | — | — | — | — | (Moqrich et al., 2005) |
| IPP | — | — | — | — | — | + | — | — | — | — | (Bang et al., 2011) |
| 4αPDD | — | — | — | — | — | — | + | — | — | — | (Watanabe et al., 2002) |
| RN 1734 | — | — | — | — | — | — | — | + | — | — | (Vincent et al., 2009) |