Table 2.
ID | RMSD (Å)a | %RefMatchb | %MolMatchc | RMSD (Å)a,d | %RefMatchb,d | %MolMatchc,d |
---|---|---|---|---|---|---|
1 (RC-33) | 0.86 | 100 | 100 | |||
2 | 1.70 | 50 | 61 | 2.30 | 50 | 61 |
3 | 1.40 | 50 | 55 | 1.82 | 50 | 55 |
4 | 2.61 | 36 | 47 | |||
5 | 2.20 | 36 | 47 | |||
6 | 1.42 | 36 | 42 | |||
7 | 0.46 | 64 | 74 | |||
8 | 2.94 | 36 | 62 | |||
9 | 1.67 | 36 | 53 | |||
10 | 2.50 | 36 | 53 | |||
11 | 2.80 | 50 | 65 | 2.89 | 50 | 65 |
12 | 2.05 | 50 | 65 | 2.16 | 50 | 65 |
13 | 2.21 | 50 | 61 | 1.50 | 50 | 61 |
14 | 1.43 | 50 | 58 | 1.46 | 50 | 58 |
15 | 0.43 | 77 | 89 | 0.86 | 77 | 89 |
16 | 1.45 | 50 | 42 | 1.07 | 50 | 42 |
17 | 0.97 | 77 | 65 | 0.69 | 77 | 65 |
18 | 1.58 | 36 | 35 | |||
19 | 0.42 | 64 | 56 | |||
20 | 1.29 | 36 | 32 | |||
21 | 2.85 | 36 | 42 | |||
22 | 0.38 | 36 | 38 | |||
23 | 2.09 | 50 | 48 | 1.94 | 50 | 48 |
24 | 0.94 | 77 | 68 | 0.83 | 77 | 68 |
25 | 1.22 | 50 | 44 | 0.82 | 50 | 44 |
26 | 1.23 | 73 | 70 | 1.98 | 73 | 70 |
27 | 1.38 | 36 | 40 | |||
28 | 0.59 | 64 | 64 | |||
29 | 2.24 | 36 | 50 | |||
30 | 0.85 | 36 | 44 | |||
31 | 1.15 | 36 | 44 | |||
32 | 1.11 | 36 | 36 | |||
33 | 2.15 | 73 | 73 | 1.78 | 73 | 73 |
34 | 2.14 | 36 | 30 | |||
35 | 0.45 | 64 | 48 | |||
36 | 3.70 | 36 | 35 | |||
37 | 4.17 | 36 | 32 | |||
38 | 2.41 | 36 | 32 | |||
39 | 1.16 | 36 | 40 | |||
40 | 0.63 | 64 | 64 | |||
41 | 0.77 | 36 | 44 | |||
42 | 0.72 | 36 | 44 | |||
43 | 2.10 | 32 | 26 | |||
44 | 1.10 | 32 | 28 | |||
45 | 1.66 | 32 | 24 | |||
46 | 0.67 | 59 | 57 | |||
47 | 1.05 | 32 | 37 | |||
48 | 2.28 | 32 | 35 | |||
49 | 2.23 | 32 | 39 | |||
50 | 0.96 | 100 | 96 | |||
51 | 0.64 | 100 | 96 | |||
52 | 1.50 | 50 | 61 | |||
53 | 1.87 | 50 | 61 | |||
54 | 1.48 | 50 | 55 | |||
55 | 1.07 | 50 | 55 | |||
56 | 2.19 | 73 | 80 | 1.96 | 73 | 80 |
57 | 2.63 | 73 | 59 | |||
58 | 2.22 | 73 | 59 | |||
59 | 1.95e | 91 | 100 | 1.98e | 91 | 100 |
60 | 1.80 | 50 | 73 | 2.54 | 50 | 73 |
61 | 2.63 | 73 | 89 | 1.52 | 73 | 89 |
62 | 3.02 | 73 | 64 | 6.97 | 73 | 64 |
63 | 2.38e | 82 | 100 | 2.51e | 82 | 100 |
64 | 2.11 | 50 | 73 | 2.58 | 50 | 73 |
65 | 2.45 | 73 | 89 | 1.01 | 73 | 89 |
66 | 2.68 | 73 | 64 | 4.26 | 73 | 64 |
67 | 2.19e | 82 | 100 | 1.98e | 82 | 100 |
68 | 0.63 | 50 | 85 | 2.96 | 50 | 85 |
69 | 2.65 | 73 | 100 | 2.73 | 73 | 100 |
70 | 3.87 | 73 | 70 | |||
71 | 6.66 | 73 | 70 | |||
72 | 2.58e | 73 | 100 | 1.49e | 73 | 100 |
73 | 2.29 | 73 | 57 | |||
74 | 2.20 | 73 | 57 | |||
75 | 4.65 | 73 | 67 | |||
76 | 4.39 | 73 | 67 | |||
77 | 2.72 | 73 | 55 | |||
78 | 2.34 | 73 | 55 | |||
79 | 1.74 | 73 | 57 | |||
80 | 2.08 | 73 | 57 |
RMSD values considering only the common chemical fragments between the docked compound and the reference compound RC-33.
%RefMatch refers to the percent of common graphs between the docked and reference compound RC-33 concerning the total number of atoms of the reference compound RC-33.
%MolMatch refers to the percent of common graphs between the docked and reference compound RC-33 regarding the total number of atoms of the docked compound.
RMSD, %RefMatch, and %MolMatch values for the S enantiomer of the compounds reported as racemic pairs.
In this case, difference in ring heavy atoms were not considered between the docked compound and the reference compound RC-33.