Table 2. Substrate Scope.
compound | R1 | R2 | yielda (%) |
---|---|---|---|
1a | 4-OMePh | c-Hex | 53 |
1b | 4-OMePh | t-Bu | 73 |
1c | 4-OMePh | 2,6-diMePh | 17 |
1d | 4-ClPh | c-Hex | 27 |
1e | 4-ClPh | t-Bu | 41 |
1f | 4-ClPh | 2,6-diMePh | 12 |
1g | Ph | c-Hex | 60 |
1h | Ph | t-Bu | 46 |
1i | Ph | 2,6-diMePh | 30 |
1j | ANT | c-Hex | 70 |
1k | ANT | t-Bu | 41 |
1l | ANT | 2,6-diMePh | 22 |
1m | t-Bu | c-Hex | 76 |
1n | t-Bu | t-Bu | 32 |
1o | t-Bu | 2,6-diMePh | 21 |
Calculated after purification.