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. Author manuscript; available in PMC: 2020 Feb 11.
Published in final edited form as: Angew Chem Int Ed Engl. 2019 Jan 16;58(7):2134–2138. doi: 10.1002/anie.201813055

Table1.

Ligand Screening for Enantioselective Arylation of Cyclopropanecarboxylic Acida,b

graphic file with name nihms-1035213-t0002.jpg
[a]

Conditions: 1a (0.1 mmol), 2a (1.5 equiv), Pd(OAc)2 (10 mol%), ligand (20 mol%), Ag2CO3 (1.5 equiv), K2HPO4 (1.5 equiv), BQ (0.5 equiv), H2O (10.0 equiv), t-BuOH (1.0 mL), 80 °C, air, 12 h.

[b]

1H NMR yields, using CH2Br2 as an internal standard. BQ = benzoquinone.