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. 2017 Nov 1;2(11):7525–7531. doi: 10.1021/acsomega.7b01542

Table 2. Synthesis of Multisubstituted Furans (3) from 2-(Aziridin-2-ylmethylene)malonate or 1,3-Dione (2) with BF3·OEt2a.

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a

Reaction conditions: 1,3-dione 2 (1.0 equiv) and BF3·OEt2 (1.05 equiv) in CH2Cl2 (0.3 M) at rt.

b

Starting ketone 2p was prepared in situ and directly converted to furan derivative 3p.