Skip to main content
. Author manuscript; available in PMC: 2019 Jul 25.
Published in final edited form as: Bioorg Med Chem. 2018 Apr 11;26(19):5270–5273. doi: 10.1016/j.bmc.2018.04.002

Table 5.

Examples of intramolecular amination in water.

graphic file with name nihms-1034553-t0007.jpg

Condition 10 mol % AgOTf, 12.5 mol % tpa, 2 equiv phIO, 0.1 M H2O, 40 °C. adr = 6.5:1 syn:anti bdr = 7.0:1 syn:anti