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. 2019 Feb 28;15(2):121–130. doi: 10.6026/97320630015121

Table 7. Comparative ADMET profile of the test ligands and the control.

Compounds Blood-Brain Barrier (BBB+/BBB-) Human Intestinal Absorption(HIA) AMES toxicity Carcinogenicity LD50 in rat
CID 126941 (Methotrexate) 0.9467 (BBB-) 0.8261 (HIA+) 0.9132 (Non AMES Toxic) Non- carcinogenic 3.4955
CID 5161 (Salsalate) 0.8946 (BBB+) 0.9161 (HIA+) 0.9731 (Non AMES Toxic) Non- carcinogenic 2.4607
CID (122677576) 0.6563 (BBB-) 0.9575 (HIA+) 0.7703 (Non AMES Toxic) Non- carcinogenic 2.6698
CID (102026478) 0.9467 (BBB-) 0.8261 (HIA+) 0.9132 (Non AMES Toxic) Non- carcinogenic 3.4955