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. 2019 Feb 28;15(2):68–78. doi: 10.6026/97320630015068

Table 7. Comparative ADMET profile of the test ligands and the control.

Blood-Brain Barrier Human Intestinal Absorption AMES Toxicity Carcinogenicity LD50 in rats
CP 690,550 (Tofacitinib) 0.9568 0.9897 0.5492 Non- carcinogenic 2.7249
Cmpd 4 0.9806 0.9958 0.584 Non- carcinogenic 2.5278
PubChem CID 76749591 0.9598 0.9956 0.5407 Non- carcinogenic 2.7101
PubChem CID 123462422 0.9631 0.9973 0.5608 Non- carcinogenic 2.7365