Table 4.
Host-derived FPR (Fpr) ligands and their classification.
Agonist | Classification | Receptor | Citation |
---|---|---|---|
CKβ 8-1 [human CCL23] | CCL23 chemokine | FPR2 | [66] |
SHAAGtide | CKβ 8-1 | FPR2 | |
Humanin | FPR2 | [98] | |
F2L | Heme binding protein | FPR2, FPR3 | [71,72,73] |
SAA | FPR2 | [90] | |
Annexin 1/ Lipocortin 1 | FPR2 | [78] | |
Ac1-25 | Annexin 1 | FPR2 | [83] |
Ac2-26 | Annexin 1 | FPR2 | [84] |
Ac9-25 | Annexin 1 | FPR2 | [85] |
Antiflammin-2 (AF-2) | FPR2 | [99] | |
Aβ-42 | Amyloid peptide | FPR2 | [60] |
D2D3 | Urokinase receptor | FPR2 | [70] |
SRSRYp | Urokinase receptor | FPR2 | |
LL-37 | Antimicrobial peptide | FPR2 | [92] |
PrP106–126 | Prion protein | FPR2 | [62] |
PACAP27 | Pituitary adenylate cyclase | FPR2, FPR1 | [63,64] |
uPAR88-92 | Urokinase receptor | FPR2 | [68] |
uPAR84-95 | Urokinase receptor | FPR2, FPR3 | [69] |
Cathepsin G | FPR1 | [100] | |
FAM3D | Chemokine-like | FPR1, FPR2 | [75] |
FAM19A4 | Chemokine-like | FPR1 | [13] |
ATLXA4 acetylsalicyclic acid-triggered | Arachidonic acid derivative | FPR2 | [101] |
Resolvin D1 (RvD1) and aspirin-triggered RvD1 | Specialized pro-resolving lipid mediator | FPR2 | [102] |
Vasoactive intestinal protein | FPR2 | [65] | |
Lipoxin-A4/Apsirin-triggered lipoxins | Fatty Acid | FPR2 | [103] |