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. 2019 Jul 12;20(14):3426. doi: 10.3390/ijms20143426

Table 4.

Host-derived FPR (Fpr) ligands and their classification.

Agonist Classification Receptor Citation
CKβ 8-1 [human CCL23] CCL23 chemokine FPR2 [66]
SHAAGtide CKβ 8-1 FPR2
Humanin FPR2 [98]
F2L Heme binding protein FPR2, FPR3 [71,72,73]
SAA FPR2 [90]
Annexin 1/ Lipocortin 1 FPR2 [78]
Ac1-25 Annexin 1 FPR2 [83]
Ac2-26 Annexin 1 FPR2 [84]
Ac9-25 Annexin 1 FPR2 [85]
Antiflammin-2 (AF-2) FPR2 [99]
Aβ-42 Amyloid peptide FPR2 [60]
D2D3 Urokinase receptor FPR2 [70]
SRSRYp Urokinase receptor FPR2
LL-37 Antimicrobial peptide FPR2 [92]
PrP106–126 Prion protein FPR2 [62]
PACAP27 Pituitary adenylate cyclase FPR2, FPR1 [63,64]
uPAR88-92 Urokinase receptor FPR2 [68]
uPAR84-95 Urokinase receptor FPR2, FPR3 [69]
Cathepsin G FPR1 [100]
FAM3D Chemokine-like FPR1, FPR2 [75]
FAM19A4 Chemokine-like FPR1 [13]
ATLXA4 acetylsalicyclic acid-triggered Arachidonic acid derivative FPR2 [101]
Resolvin D1 (RvD1) and aspirin-triggered RvD1 Specialized pro-resolving lipid mediator FPR2 [102]
Vasoactive intestinal protein FPR2 [65]
Lipoxin-A4/Apsirin-triggered lipoxins Fatty Acid FPR2 [103]
HHS Vulnerability Disclosure