. Author manuscript; available in PMC: 2020 Aug 1.

Published in final edited form as: FEBS Lett. 2019 Jun 18;593(15):2069–2078. doi: 10.1002/1873-3468.13474

Table:2.

IC50(μcm) for ChTS and hTSa.

Compound	ChTS IC₅₀	hTS IC₅₀	Fold-Selectivity
1^b	0.38 ± 0.04	1.8 ± 0.5	5
2	9.8 ± 0.6	0.6 ± 0.2	16
Fold-Stereospecificity	26	3

SD from triplicate measurement.

Results from reference [11]