a) qPCR analysis of ABCA1 mRNA in THP-1
macrophages transfected with control (ctrl) or CHROME-targeting
GapmeRs. Data are the mean ± SEM of 3 independent experiments. (b)
Western blot of ABCA1 and HSP90 (internal control) protein in THP-1 macrophages
transfected with control (ctrl) or CHROME-targeting GapmeRs.
Molecular weight marker is shown at right. Data are representative of 3
independent experiments. c, Measurement of cholesterol efflux to
exogenous apoA-1 in THP-1 macrophages transfected control (ctrl) or
CHROME-targeting GapmeRs. Data are the mean ± SEM of
4 independent experiments. d-e, Activity of (d)
ABCA1-3’UTR and (e)
OSBPL6-3’UTR luciferase reporter genes in HEK293T cells
expressing empty vector (EV), wild type CHROME-7
(CHROME-7WT), or CHROME-7 with
its miR-33, miR-27b and miR-128 binding sites mutated
(CHROME-7MUT) following treatment with control
miR, miR-27b or miR-33 mimics. Data are the mean ± SEM of 3 biological
replicates from a single experiment. Data are representative of 3 independent
experiments. f, qPCR analysis of miR-27b, miR-33 and miR-128 target
genes regulating cholesterol efflux in THP-1 macrophages stably expressing empty
vector, CHROME-7WT or
CHROME-7MUT. Data are the mean ± SEM of 3
experiments. g, Measurement of cholesterol efflux to apoA-1 in
THP-1 macrophages stably expressing empty vector,
CHROME-7WT or
CHROME-7MUT. Data are the mean ± SEM of 3
experiments. h, Representative images of Nile Red stained lipid
droplet accumulation in acetylated LDL treated THP-1 macrophages stably
expressing empty vector, CHROME-7WT or
CHROME-7MUT. Cells were stained with DAPI (blue)
to visualize nuclear DNA. i, qPCR analysis of miRNA levels in THP-1
cells stably expressing empty vector, CHROME-7WT or
CHROME-7MUT. miR-16 is included as a negative
control. Data are the mean ± SEM of 3 experiments. P-values were
calculated using a two-tailed student’s t-test. *P≤0.05,
**P≤0.01, ***P≤0.001.