S2.
Anticancer drugs comprising the small compound library for the screen
| Table of compounds tested from the combined TDI Extended Oncology Drugs Library (ODL) and the NCI Developmental Therapeutics Program (DTP) Approved Oncology Drug Library. | ||||
| (5Z)-7-Oxozeaenol | Bleomycin | FK 506_Tacrolimus | Mitomycin C | Rapamycin (sirolimus) |
| (R)-Flurbiprofen (Tarenflurbil) | BMS-754807 | FK-866 HCl_Daporinad | Mitotane | RD162 |
| 1-methyl-D-tryptophan, 95% | BMS-911543 | Floxuridine | Mitoxantrone | RDEA119_Refametinib |
| 17-AAG (Tanespimycin, Geldanamycin) | Bortezomib | Fludarabine | MK-0752 | Ridaforolimus |
| 17-DMAG (Alvespimycin) | Bosutinib | Fluorouracil | MK-2206 | Rofecoxib (Vioxx) |
| 2-methoxyestradiol (Panzem) | Brivanib | Flutamide | MK-4827, HCl salt | Romidepsin |
| 4-hydroxytamoxifen | Busulfan | Fulvestrant | MK1775 | Roscovitine_Selicilib |
| Abitrexate/Methotrexate | Cabazitaxel | Galiellalactone | MLN4924 | S-trityl-L-cysteine, 40 mM |
| ABT-199 | CAL-101 | GDC-0068 | MLN8237_Alisertib | SB 743921 |
| ABT-263 (Navitoclax) | Camptothecin | GDC-0941_Pictilisib | Motesanib Di phosphate (AMG-706) | Simvastatin |
| ABT-751 | Canertinib | GDC-0980 | Nelarabine | Sorafenib |
| ABT-869_Linifanib | Capecitabine | Gefitinib | Nilotinib | Sotrastaurin |
| ABT-888 (Veliparib) | Carboplatin | Gemcitabine HCl | Nilutamide | SR1 HCl |
| AC220_Quizartinib | Carfilzomib | Goserelin acetate | Nitrogen mustard | Stattic |
| Acrichine | Carmustine | GSK 269962 | Nutlin-3 | Streptozocin |
| AG-014699_Rucaparib | Celecoxib | GSK 650394 | NVP-AUY922 | Sunitinib |
| Allopurinol | CHIR-258 (Dovitinib) | GSK1120212_ Trametinib | NVP-BEZ235_Dactolisib | TAK-733 |
| Altretamine | Chlorambucil | GSK2126458 | NVP-BGJ398 | TAK-901 |
| Amifostine | Chloroquine diphosphate | GSK2636771 | NVP-LDE225 (Diphosphate salt) | Tamoxifen citrate |
| Aminoglutethimide | CHR 2797_Tosedostat | HA-1077 (Fasudil) | Obatoclax Mesylate (GX15-070) | Tandutinib |
| Aminolevulinic acid | CI-994_Tacedinaline | Homoharringtonine | Olaparib | Tasocitinib_Tofacitinib |
| Amonafide | Cisplatin aq | Hydroxyurea | OSI-027 | Temozolomide |
| Anagrelide | Cladribine | I-BET151 (GSK1210151A) | OSI-906_Linsitinib | Teniposide |
| Anastrozole | Clafen (Cyclophos-phamide, Endoxan) | Idarubicin HCl | Oxaliplatin | Tetramisole HCl |
| AP24534 (Ponatinib) | Clofarabine | Ifosfamide | PAC-1 | TGX-221 |
| ARQ 197_Tivantinib | Clomifene citrate | Imatinib | Paclitaxel | Thalidomide |
| ARRY-162_MEK-162 | CPI-613 | Imiquimod | Panobinostat | Thio-TEPA |
| Arsenic(III) oxide | Crenolanib | INCB018424 (free base, Ruxolitinib) | Pazopanib | Thioguanine |
| AS703026_Pimasertib | Crizotinib | Indibulin | PCI-32765_Ibrutinib | Thiotepa |
| Aspirin (Acetylsalicylic Acid) | CUDC-101 | Iniparib (BSI-201, IND-71677) | PD-0332991 | Tipifarnib (Zarnestra) |
| AT 101 | Cyclophosphamide | INK128 | Pemetrexed | Topotecan HCl |
| AT-406 | CYT-387_Momelotinib | Irinotecan | Pentostatin | Toremifene citrate |
| AT9283 | Cytarabine HCl | Ixabepilone | Perifosine aq/PBS | Tretinoin |
| Atorvastatin Ca | Dabrafenib Mesylate | JNJ 26854165 (Serdemetan) | PF 431396 | Triethylenemelamine |
| Auranofin | Dacarbazine | JNJ_26481585_Quisinostat | PF 477736 | Tubacin |
| AV-951 (Tivozanib) | Dacomitinib (monohydrate) (PF-00299804) | KX2-391 | PF-04691502 | Tubastatin A HCl |
| AVN944 | Dactinomycin | Lapatinib, di-p-toluenesulfonate salt | PF-04708671 | UCN-01 |
| Axitinib | Dasatinib | Lasofoxifene | PF-2341066 (Crizotinib) | Uracil mustard |
| AZ 3146 | Daunorubicin HCl | Lenalidomide | PF-3845 | Valproic acid |
| Azacitidine | DCC-2036_Rebastinib | Lestaurtinib | PF4800567 hydrochloride | Valrubicin |
| AZD 7762 hydrochloride | Decitabine | Letrozole | PF670462 | Vandetanib |
| AZD1152-HQPA | Decitabine (Dacogen) | Lomeguatrib | PHA-739358 (Danusertib) | Varespladib |
| AZD1480 | Deferoxamine mesylate | Lomustine, CCNU | PIK-75 HCl | Vatalanib |
| AZD2014 | Dexamethasone (Decadron) | LY 333531 mesylate- Ruboxistaurin | Pilocarpine | Vemurafenib |
| AZD4547 | Dexrazoxone | LY2157299 | Pipobroman | VER 155008 |
| AZD6244 (Selumetinib) | Dinaciclib (SCH727965) | LY2228820 (CP868569) | PKC412_Midostaurin | Vinblastine sulfate |
| AZD8055 | Docetaxel | LY2603618_Rabusertib | Plerixafor | Vincristine Sulfate (Oncovin) |
| BAY 73-4506_Regorafenib | Doxorubicin | LY2784544_Gandotinib | Plicamycin | Vinorelbine tartrate |
| Belinostat (PXD101) | Doxorubicin HCl | Masitinib | PLX4032_Vemurafenib | Vismodegib |
| Bendamustine HCl | EMD1214063 | MDV3100_Enzaluamide | Pralatrexate | Vorinostat |
| Bexarotene | Entinostat | Megestrol acetate | Pravastatin | VX-11e |
| BI 2536 | Enzastaurin | Melphalan | Prednisolone | XAV-939 |
| BI 6727_Volasertib | Epothilone B (Patupilone) | Mercaptopurine | Prednisone | XL-147 |
| BIBF 1120_Nintedanib | Erlotinib HCl | Metformin
hydrochloride aq |
Prima-1 Met | XL184_Cabozantinib |
| BIBW2992 (Tovok)_Afatinib | Estramustine sodium phosphate | Methotrexate | Procarbazine | XL880 (Foretinib) |
| Bicalutamide | Etoposide | Methoxsalen | PX-866_Sonolisib | YM155 |
| BIIB021 | Everolimus | Methylprednisolone | Quinacrine HCl | Zolendronic acid |
| Bimatoprost | Exemestane | MGCD-265 | R406_Tamatinib | ZSTK474 |
| BIRB 796 (Doramapimod) | FG-4592 | MGCD0103_Mocetinostat | RAF265 | |
| BKM-120_Buparlisib | Finasteride | Mithramycin A | Raloxifene HCl | |