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. 2019 Aug 15;4(9):14151–14154. doi: 10.1021/acsomega.9b02144

Table 1. Receptor Binding Affinity^a.

antagonist	D₂K_I (nM)	5-HT₇ K_I (nM)
amisulpride (S)	n.d.	900 ± 1300
amisulpride (rac)	1.1 ± 0.12	44 ± 3
amisulpride (R)	n.d.	22 ± 1.5
LB-102	0.82 ± 0.02	31 ± 1
LB-103	0.4 ± 0.04	>1000
LB-104	14.4 ± 2.2	15.6 ± 0.9

^a

n.d. not determined.