Table 3.
Parameters | AIF in 25% Cremophor EL®/EtOH Solution | AIF-Loaded mPEG-b-PLA Micelle |
---|---|---|
AUC a (min·μg·mL−1) | 326 ± 168 | 876 ± 103 * |
C0 b (μg·mL−1) | 1.89 ± 0.63 | 7.86 ± 1.79 |
CLt c (mL·kg−1·min) | 94.6 ± 56.1 | 23.1 ± 2.7 |
Vd d (mL·kg−1) | 13903 ± 5274 | 2940 ± 867 |
BA e (%) | 100 ± 51 | 269 ± 18 * |
a AUC, area under the curve; b C0, plasma concentration at time 0; c CLt, total clearance; d Vd, volume of distribution; BAe, bioavailability, * p < 0.05.