Table 2. Scale factors used to simulate pharmacological manipulation with Moxifloxacin.
IC50 = 86.2 μM Hill slope = 0.94 |
Moxifloxacin | IC50 = 173 μM Hill slope = 1 |
IC50 = 1112 μM Hill slope = 1 |
---|---|---|---|
Scale factor gKr | Concentration [μM] | Scale factor gCaL | Scale factor gNa |
0.25 | 277.4 | 0.38 | 0.80 |
0.5 | 86.2 | 0.67 | 0.93 |
0.9 | 8.32 | 0.95 | 0.993 |
0.95 | 3.76 | 0.979 | 0.997 |