Skip to main content
. 2019 Sep 20;92(3):369–383.

Table 2. Estimate of selectivity index for natural product isolates.

Compounds IC50Toxoplasma gondii (µg/mL) IC50 HFF cells (µg/mL) Selectivity Index (SI)
Rhapontin 1.22 20.05 16.38 SI >1
Homobutein 4.43 68.28 15.41 SI >1
Sulfuretine 0.68 8.20 12.10 SI >1
Arbutin 17.20 84.23 4.90 SI >1
Butein 2.12 7.92 3.74 SI >1
Naringenin 3.03 9.20 3.03 SI >1
Narasin 0.74 2.09 2.84 SI >1
Stachydrine.HCl 4.40 10.41 2.36 SI >1
Shikonin 3.96 5.81 1.47 SI >1
Hesperitine 13.66 12.42 0.91
Lasalocid A 1.61 1.46 0.90
Ochratoxin A 11.33 9.63 0.85
Radicicol 4.90 2.58 0.53
Cephaeline.HBr 0.95 0.45 0.47
Menadione 44.70 17.93 0.40
Peruvoside 0.37 0.11 0.30
Sulfadiazine 185.20 53.35 0.29
Mitomycin C 1.87 0.44 0.24
Gitoxigenin 2.59 0.62 0.24
Pyrimethamine 205.60 42.16 0.21
Strophantidin 1.30 0.19 0.15
Diacetoxyscirpenol 0.62 0.05 0.08
Tubericidin 0.46 0.02 0.04
Capsiacin ND 9.69 ND
Curcumin ND ND ND
Resveratrol 1.03 ND ND
Genistin 5.46 ND ND
Eriodictyol ND ND ND
Andrographolide 388.10 ND ND
Syringetine-3-glucoside 16.64 ND ND
Piperine 1.71 ND ND
Aloe-emodine 8.14 ND ND
Neohesperidin ND ND ND
5,6-Dehydrokawain 4.22 ND ND
Betulin 224.40 ND ND
Lavendustin A 37.45 ND ND
Gelsemine.HCl 89.29 ND ND

*ND – Not determined.