Table 3. Single agent dose response IC50s at 24-hours and 96-hours after treatment, ± standard error of the mean.
Tx | A673 | TC32 | Top Concentration | Cmax (ng/ml) | ||
---|---|---|---|---|---|---|
Day 2 | Day 5 | Day 2 | Day 5 | |||
MTIC | 18889 ± 3240 | 18915 ± 3672 | 15547 ± 7867 | 9447 ± 4045 | 250 | 276 |
SN38 | 40 ± 33 | 0.77 ± 0 | 4.0 ± 0.5 | 2.6 ± 0.2 | 4 | 30 |
SP2509 | 4222 ± 863 | 1171 ± 212 | 2375 ± 221 | 1238 ± 89 | 1000 | 3000 |
Vincristine | 0.73 ± 0.25 | 0.79 ± 0.03 | 6.2 ± 1.4 | 2.0 ± 0.3 | 1 | 40 |